Melatonin - Less is More
MIT scientists confirm that melatonin is an effective sleep aid for older insomniacs and it appears that only a small dose of melatonin (about 0.3 milligrams) is necessary for a restful effect. Taken in that quantity, melatonin not only helps people fall asleep, but also makes it easier for them to return to sleep after waking up during the night. However, the amount in most melatonin products on the market ranges between 1 to 5 mg. At this high dose, tolerance can develop and the melatonin receptors in the brain become unresponsive. Thereafter, melatonin becomes less effective.
    

Newsletter /  FAQs / Personal Stories / Dr. Sahelian /  Order Form

Melatonin: Nature's Sleeping Pill

The Right Dose of Melatonin for Sleep

After treating more than 200 patients with melatonin, surveying hundreds more, and informally talking to thousands of users, we are convinced that, until we learn more, it's best not to take melatonin on a daily basis. The following are some of our concerns:

1) Tolerance develops in some people when melatonin is used every night. After a few weeks some find that melatonin is not inducing or maintaining sleep as well as it did in the past. To avoid the creeping up of tolerance, melatonin should be used at most every other night, or preferably every third night. The dose used should be the lowest amount that works, such as 1 mg or less. Some users find that a dose as little as 0.2 mg can induce sleep. It is ok to occasionally take a high dose such as 5 or 10 mg if needed. Melatonin is not toxic at high doses when used infrequently.

2) Tiredness, low mood, or fatigue can develop when people use melatonin every night, especially in doses more than 2 or 3 mg. Some people feel sleepy the next day with the wish to take naps.

3) We still don't know the long-term effects on the immune and hormonal systems of chronic melatonin use. Also, high doses of melatonin used regularly could possibly inhibit sex drive and inhibit the function of gonads (testicles and ovaries).

I'm 40 years old and I'm currently using 0.5 mg of melatonin about twice a week. Not only does melatonin provide me with a deep sleep, but there seems to be a carry over effect into following nights. The effect of taking it one night seems to influence my sleep positively for another night or two. Many users find the same: they feel better, have a better mood and more energy.

I also take melatonin with the hopes of living longer. The effect of melatonin on longevity could be due to many factors, and let's briefly discuss three of them:

1) Deep Sleep. The positive influence of melatonin on deep, restorative sleep could alone account for a longer life span.

2) As an antioxidant. The advantage of melatonin over other antioxidants is that it is both water and fat soluble, meaning it goes into almost all cells and all parts of the body. Melatonin's disadvantage is that it has a short half-life and it's antioxidant benefits may only last overnight, as opposed to vitamin E, which is stored in tissues and protects all day long.

3) Immune system improvement. Interestingly, many people report that since they've been on melatonin, they don't catch colds and infections as much as they used to. These stories are, of course, anecdotal, and we don't have any published human studies on the influence of melatonin on the immune system in the long-term.

Chapter One

Melatonin: A Supplement for the Future? or Tonight?

Discusses the controversy, safety issues, and effectiveness.

Chapter Two

From Cradle to Rocking Chair-Melatonin Throughout Life

Includes a graph of declining levels throughout life.

Chapter Three

Dreams Like You Never Dreamed

Melatonin has the Chemical Structure Similar to Tryptamine Hallucinogens

Dr. Sahelian Proposes that Dreams may be Hallucinogenic Experiences

Chapter Four

Melatonin and Longevity

Life Span Extension in Animals

A Powerful Antioxidant

Immune Enhancement

An Honest Appraisal of Melatonin's Influence on Longevity

Chapter Five

Take Two Melatonin's and Call Me in the Morning

What Dosage is Best?

When is the Best Time to Take Melatonin?

Is Melatonin Addictive?

What About Tolerance?

Are Their Withdrawl Symptoms?

Chapter Six

Uses of Melatonin: Insomnia, Jet Lag, Shift Work, Mood Elevation

Chapter Seven

The Circadian Cycle

The Pineal Gland

Hibernation

Daily Rhythms

Chapter Eight

The Science of Sleep

The Lessons from the Blind

The Stages of Sleep

Chapter Nine

Twenty Tips to Forty Winks

How to Sleep Deep

Chapter Ten

Melatonin and the Future

To Lower Cholesterol Levels

To Treat Prostate Gland Enlargement

Treating Osteoporosis, Cancer, Epilepsy, Improving Immunity

For Heart Disease and to Prevent Cataracts

Appendix

The Chemistry of Melatonin

Personal Stories of Melatonin Users